Products
HBT1 foda (489408-02-8) bidiyo
HBT1 foda (489408-02-8) Bayanin Base
sunan | HBT1 foda |
CAS | 489408-02-8 |
tsarki | 98% |
Chemical name | 2-(((5-Methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl)acetyl)amino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide |
nufin abu ɗaya ne | HBT1; HBT-1; Farashin HBT1 |
kwayoyin Formula | C16H17F3N4O2S |
kwayoyin Weight | 386.39 |
Ƙaddamarwa Point | / |
InChI Key | PHLXSNIEQIKENK-UHFFFAOYSA-N |
Form | foda |
Appearance | fararen fata |
Rabin Rayuwa | / |
solubility | DMSO: 2 MG / ML, bayyana |
Storage Yanayin | 0 - 4 C don gajere (kwanaki zuwa makonni), ko -20 C na dogon lokaci (watanni). |
Aikace-aikace | Amintaccen mai karɓar AMPA |
Takardar Gwaji | Ya Rasu |
HBT1 foda (489408-02-8) Babban bayanin
HBT1 foda shine mai karɓar mai karɓar AMPA tare da ƙananan tasirin azaba, yana guje wa amsa mai kama da kararrawa a cikin aikin BDNF na vitro. Amfani ne na AMPA-R [alpha-amino-3-hydroxy-5-methyl-4-isoxazole-propionic acid (AMPA)] wanda ke haifar da samar da kwayar cutar da ke haifar da kwakwalwa (BDNF) kuma tana nuna tasirin tashin hankali a matakin farko ƙwayoyin cuta HBT1 yana ɗaure ga yankin AMPA-R mai ɗaukar ligand a cikin hanyar dogara da glutamate.
HBT1 foda (489408-02-8) Tunani
[1] Kunugi A, Tajima Y, Kuno H, Sogabe S, Kimura H. HBT1, Novel AMPA Receptor Potentiator with Lower Agonistic Effect, Guji Amsa Kirar Bell a cikin Injin Vitro BDNF. J Pharmacol Mai Magana. 2018 Mar; 364 (3): 377-389. Doi: 10.1124 / jpet.117.245050. Epub 2018 Jan 3. An buga PMID: 29298820.
Labarai masu amfani
blog
Tuntube mu
Game damu
Our Products
- Nootropics foda
- Alzheimer ta cutar
- Rakiya
- kari
- Aniracetam Review: Shin wannan Nootropic foda yana da kyau a gare ku?
- Glycine Propionyl-L-Carnitine (GPLC): Mafi kyawun Forarshe don Gina Jiki
- Mafi kyawun Bitamin C 3-O-Ethyl-L-ascorbic Acid a Amfani da Kayan shafawa
- Mafi kyawun Jagora na Nootropic: Duk Abubuwan da kuke Bukatar Ku sani [Shekaru 5 na Kwarewa]
- PQQ foda (72909-34-3)
- Nmn foda (1094-61-7)
- Aniracetam foda (72432-10-1)/li>
- Glucoraphanin foda 30% (21414-41-5)