Products
THM foda (1224690-84-9) bidiyo
THM foda (1224690-84-9) Base Information
sunan | Tianeptine hemisulfate monohydrate (THM) foda |
CAS | 1224690-84-9 |
tsarki | 98% |
Chemical name | Tianeptine hemisulfate monohydrate; 1224690-84-9; Heptanoic acid, |
nufin abu ɗaya ne | Tianeptine hemisulfate monohydrate 1224690-84-9 7 - ((3-Chloro-6-methyl-5,5-dioxido-6,11-dihydrodibenzo [c, f] [1,2] thiazepin-11-yl) amino) tarin kwayoyin acid mai narkewa tare da acid na sulfuric (2: 1) bushewar ruwa Sinadarin Tianeptine; Tianeptine-d4 BCP30653 |
kwayoyin Formula | C42H56Cl2N4O14S3 |
kwayoyin Weight | 1008.01 |
Ƙaddamarwa Point | 1800 ℃ |
InChI Key | KVVMXNNJBVTOSX-UHFFFAOYSA-N |
Form | foda |
Appearance | Farin crystalline foda |
Rabin Rayuwa | Rashin sani |
solubility | Creetly soluble A cikin ruwa da methanol da dichloromethane |
Storage Yanayin | Tianeptine hemisulfate monohydrate foda yana da kwanciyar hankali na akalla shekaru hudu lokacin da aka adana shi kuma ba'a yanke shi a −20 ° C ba. |
Aikace-aikace | Anti-ulcer da anti-kwayoyin mallaka. Labarin |
Takardar Gwaji | Ya Rasu |
THM foda (1224690-84-9) Babban bayanin
Ana amfani da sulfate na Tianeptine da farko a cikin lura da rikicewar damuwa, kodayake ana iya amfani da shi don magance asma ko ciwo na hanji. Chemically shi ne mai tricyclic antidepressant (TCA), amma yana da kaddarorin magunguna daban-daban fiye da TCAs na yau da kullun kamar yadda bincike na kwanan nan ya nuna cewa tianeptine yana haifar da tasirin antidepressant ta hanyar canji na ayyukan mai karɓar glutamate (watau masu karɓar AMPA da masu karɓar NMDA) da sakin BDNF, bi da bi shafi na tsarin filastik.
Tianeptine sulfate yana da antidepressant da anxiolytic (anti-damuwa) kaddarorin da ke da dangin rashin kwantar da hankali, anticholinergic da cututtukan cututtukan zuciya, don haka yana ba da shawarar cewa ya dace musamman don amfani a cikin tsofaffi da cikin waɗanda ke biye da shan giya; irin waɗannan mutane na iya zama masu kula da illolin magungunan psychotropic. Sakamakon da aka samu kwanan nan yana nuna yuwuwar ƙwanƙwasawa (anti-seizure) da analgesic (painkilling) aikin tianeptine ta hanyar sauƙaƙe ko canjin yanayin adenosine A1 masu karɓa (kamar yadda masu adawa da wannan mai karɓa za su iya katange sakamakon.
THM foda (1224690-84-9) Tarihi
Tsarin Tianeptine sulfate (Tianeptine Hemisulfate Monohydrate (THM)) an rarrabe shi azaman mai zaɓin mai haɓaka ƙwaƙwalwar serotonin (SSRE) wanda aka yi amfani dashi don magance rashin damuwa. Tianeptine an haɓaka shi a Faransa a cikin 1960s kuma anyi amfani dashi a ƙarshen ƙarshen 2000s. Akwai sulfate sulfate, soda na Tianeptine, da acid acid Tianeptine.
An tsara shi azaman mai zaɓin kayan haɓaka na serotonin reuptake (SSRE) wanda aka yi amfani dashi don magance ɓacin rai. Tianeptine an haɓaka shi a Faransa a cikin 1960s kuma anyi amfani dashi a ƙarshen ƙarshen 2000s. Akwai sulfate sulfate, soda na Tianeptine, da acid acid Tianeptine.
THM foda (1224690-84-9) Hanyar Nawa
Ba kamar yawancin antidepressants ba, Tianeptine yana da ƙananan tasirin illa; Tianeptine yana nuna alƙawari a matsayin madadin masu maganin ƙwaƙwalwar gargajiyar gargajiya da halayensu na jaraba da jerin abubuwan da ke haifar dasu.Yayin da yawancin masu amfani da maganin ba sa zagi ko amfani da magungunan, an ba su umarnin, wannan ba ya magana da sauran jama'a. . Magungunan kwantar da hankali sanannen aiki ne na haɗari. Ga mutanen da ba sa buƙatar su, shan irin waɗannan ƙwayoyi na iya zuwa da illoli masu yawa da yawa da kuma haɗarin kayan maye. Tianeptine na iya zama madadin mafi aminci ga yawancin antidepressants da ke kasuwa a yau. Lissafin cututtukan da ke tattare da su ƙananan ne kuma ana iya jure su, sun haɗa da bacci, bushe-bushe, rashin bacci, jiri, jiri, maƙarƙashiya, ƙarancin hawan jini, kuma wasu marasa lafiya suna kwatanta mafarkai masu ban mamaki.
THM foda (1224690-84-9) Aikace-aikace
Magungunan Tianeptine don magance cututtukan kwakwalwa, bincike sun nuna cewa tianeptine ba kawai kyakkyawan sakamako na antidepressant da halayen haɗari sun kasance ƙasa da ƙananan magungunan maganin tricyclic na al'ada, kusan babu mummunar tasiri akan tsarin jijiyoyin jini, jini, hanta da aikin koda ba a cutar da su ba. , kuma ba ni da nutsuwa. Tianeptine ba kawai tasiri bane don bacin rai da nakasa mai narkewa, rashin shan giya da bacin rai bayan shan giya shima yana da tasiri. Amfani da na dogon lokaci na iya hana sake komawa
THM foda (1224690-84-9) researcharin bincike
Anyi nazarin Magnesium ta beraye don jinkirta farawa da ci gaban cututtukan cataract.
Hakanan ana amfani da Tianeptine don magance rikicewar damuwa, asma har ma da rashin damuwa na hanji.
Kimiyya A bayan Sa:
wannan tambaya ce mai ruɗi saboda Tianeptine sulfate shine sabon fili wanda ke buƙata, kuma ya cancanci, ƙarin kudaden da aka saka a ciki don gwaji.
Abin da muka sani shi ne cewa Tianeptine Sulfate yana da alaƙa da Tianeptine Sodium, kuma yana aikatawa sosai. wannan ya faru ne saboda bambancin tsarin sunadarai, kamar yadda za'a iya gani a adadi ta hannun dama.
ga waɗanda daga cikinku suka saba da Tianeptine Sodium, ƙila ku san shi a ƙarƙashin sunan kasuwanci & lsquo; Coaxil 'ta hanyar Turai da Asiya ko kuma & lsquo; Stablon 'da & lsquo; Tatinol 'ta Latin Amurka. a halin yanzu an yarda dashi don amfani da lafiya a ƙasashe 20.
Abin mamaki, kodayake, masana kimiyya ba su da tabbaci 100% game da yadda Tianeptine yake a zahiri & lsquo; yana aiki. Tunanin farko shine cewa yayi aiki ne a matsayin mai Ingantaccen Serotonin Re-absorption Enhancer (SSRE) duk da haka binciken da aka yi kwanan nan ya nuna cewa ainihin lokacin ba shi da tasiri akan tsarin mulkin ƙasa wanda zai iya inganta matakan serotonin.
Sabbin ka'idoji game da aikin Tianeptine azaman maganin rigakafi ta hanyar canza ayyukan mai karɓar glutamate kai tsaye da kuma sakin BDNF (ƙwaƙwalwar ƙwaƙwalwar ƙwaƙwalwar ƙwaƙwalwar ƙwaƙwalwar ƙwaƙwalwa) wanda zai iya jujjuya yanayin jijiyoyin jiki.
akwai kuma wani sabon bincike a cikin Yulin 2014 wanda ya gano cewa Tianeptine ita ce mai azabar kai tsaye na Masu karɓar Mu da Delta Opioid. tunda ana alakanta masu karɓa na Mu-Opioid zuwa tasirin euphoric, wannan an ba da shawarar a matsayin dalili na aikin Tianeptine a matsayin mai hana tashin hankali.
THM foda (1224690-84-9) Tunani