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Nooglutyl foda (112193-35-8) bidiyo
Nooglutyl foda (112193-35-8) Labarin Base
sunan | Nooglutyl foda |
CAS | 112193-35-8 |
tsarki | 98% |
Chemical name | N - [(5-Hydroxy-3-pyridinyl) carbonyl] -L-glutamic acid N- (5-hydroxynicotinoyl) -L-glutamic acid N- (5-Hydroxymethyl-pyridin-2-yl) -2,2-dimethyl-propionamide ; nooglutil |
nufin abu ɗaya ne | nooglutil;N-[(5-Hydroxy-3-pyridinyl)carbonyl]-L-glutamic acid;N-[(5-Hydroxypyridin-3-yl)carbonyl]-L-glutamicacid;ONK-10;L-GlutaMic acid, N-[(5-hydroxy-3-pyridinyl)carbonyl]-;Nooglutyl |
kwayoyin Formula | C11H12N2O6 |
kwayoyin Weight | 268.22 g / mol |
Ƙaddamarwa Point | N / A |
InChI Key | XFZGYOJFPGPYCS-QMMMGPOBSA-N |
Form | m |
Appearance | Farar lafiya foda |
Rabin Rayuwa | 30 minti zuwa 3 hours |
solubility | kadan soluble a cikin ruwa da kuma ethanol. |
Storage Yanayin | Adana a cikin sanyi mai bushe da bushe, an kiyaye shi daga danshi da haske mai ƙarfi ko zazzabi mai zafi. |
Aikace-aikace | An yi amfani da shi a cikin magani, kayayyakin kiwon lafiya, abinci, abin sha, kayan shafawa, abubuwan nazarin halittu da sinadarai da sauran masana'antu. |
Takardar Gwaji | Ya Rasu |
Nooglutyl foda (112193-35-8) Babban bayanin
Nooglutyl wakili ne na kwayar halitta wanda ake karantawa a Cibiyar Nazarin Magungunan Magunguna, Kwalejin Kimiyyar Kiwon Lafiya ta Rasha a matsayin maganin cutar amnesia. A cikin sifofin dabbobi, yana da nau'ikan tasirin tsarin juyayi na tsakiya.
Gwaje-gwaje a kan berayen suna nuna cewa nooglutyl yana nuna alamomi masu karewa-kariya masu kariya kuma ta wurin aikin antimotion ba ya samuwa a ƙarƙashin masu tsaron gida na musamman, irin su scopolamine da diprazine. Nazarin ilimin electrophyysiological a kan garuruwa ya nuna cewa nooglutyl ya canza aiki mai ban sha'awa a 80% na ƙananan ƙananan ƙwayoyin cuta (yankin somatosensory I da yanki na 5 na ɓangaren ƙungiyar tarayya) da kuma mummunar tasirin da lalacewa ta hanyar motsi motsi: kunna aiki na ɗaya na zone na somatosensory I da kuma hanawa neuron amsa zuwa somatic stimulation. An kiyasta wannan kayan aikin shiri don samar da asali na tasirin antimotion.
Nooglutyl foda (112193-35-8) Tarihi
Nooglutyl shine nootropic Wakilin da aka yi karatu a Cibiyar Nazarin Magunguna, Kwalejin Kimiyyar Kiwon Lafiya ta Rasha a matsayin yuwuwar magani ga amnesia. A cikin dabbobin dabba, yana da tasirin tsarin jijiyoyin jiki iri -iri.
Nooglutyl foda (112193-35-8) Hanyar Neman Aiki
Gwaje-gwaje a kan berayen suna nuna cewa nooglutyl yana nuna alamomi masu karewa-kariya masu kariya kuma ta wurin aikin antimotion ba ya samuwa a ƙarƙashin masu tsaron gida na musamman, irin su scopolamine da diprazine. Nazarin ilimin electrophyysiological a kan garuruwa ya nuna cewa nooglutyl ya canza aiki mai ban sha'awa a 80% na ƙananan ƙananan ƙwayoyin cuta (yankin somatosensory I da yanki na 5 na ɓangaren ƙungiyar tarayya) da kuma mummunar tasirin da lalacewa ta hanyar motsi motsi: kunna aiki na ɗaya na zone na somatosensory I da kuma hanawa neuron amsa zuwa somatic stimulation. An kiyasta wannan kayan aikin shiri don samar da asali na tasirin antimotion.
Nooglutyl foda (112193-35-8) Aikace-aikacen
Nooglutyl shine a nootropic Ana nazarin wakili a Cibiyar Nazarin Magungunan Magunguna, Kwalejin Kimiyyar Kiwon Lafiya ta Rasha a matsayin yuwuwar magani ga amnesia.A cikin dabbobin dabba, yana da tasirin tsarin jijiyoyin jiki iri -iri.
Nooglutyl foda (112193-35-8) Tunani
- Flekhter, Oxana B. (2000). "Nooglutil, Kwalejin Kwalejin Kimiyya ta Rasha". Sanarwa ta yanzu a cikin Magungunan Binciken Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Tsarin Magunguna 2 (4): 491–
- V. Yasnetsov; VA Pravdivtsev; VM Popov; TA Voronina; NM Kiseleva; SB Kozlov (Mayu 1995). "Tasirin Antimotion na Nooglutyl da Tsarin Neuronal". Sanarwa game da Gwajin Biology da Magani. 119 (5): 515-516. Doi: 10.1007 / BF02543440. PMID 7579248. An dawo da shi 2011-02-08.
- Voronina, TA; Borlikova, GG; Garibova, TL; Proskuryakova, TV; Petrichenko, OB; Burd, SG; Avakyan, GN (2002). "Tasirin nooglutil akan cutar ciwon benzodiazepine da ɗaukar 3H-spiperone tare da masu karɓar D2 a cikin rat striatum". Sanarwa game da ilmin gwaji da magani. 134 (5): 448–